Enitociclib
Tier C — Watch / tradeEnitociclib
Targets：CDK9, PTEFb
Indications (approved)：Non-Hodgkin lymphoma, Lymphoma, Haematological malignancy, Neoplasm, 里氏综合征, Chronic lymphocytic leukaemia
Regional status
Synthetic routes & intermediates1 routes
Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.
| Code | CAS No. | Intermediate |
|---|---|---|
| BAY-1251152 | 1610358-53-6 | ((2-((5-fluoro-4-(4-fluoro-2-methoxyphenyl)pyridin-2-yl)amino)pyridin-4-yl)methyl)(imino)(methyl)-l6-sulfanone |
| BAY-1251152-001 | 179899-07-1 | (4-fluoro-2-methoxyphenyl)boronic acid |
| BAY-1251152-002 | 884494-49-9 | 2-chloro-5-fluoro-4-iodopyridine |
| BAY-1251152-003 | 1602486-03-2 | 2-chloro-5-fluoro-4-(4-fluoro-2-methoxyphenyl)pyridine |
| BAY-1251152-004 | 179554-98-4 | 4-((methylthio)methyl)pyridin-2-amine |
| BAY-1251152-005 | 1602486-04-3 | 5-fluoro-4-(4-fluoro-2-methoxyphenyl)-N-(4-((methylthio)methyl)pyridin-2-yl)pyridin-2-amine |
| BAY-1251152-006 | 354-38-1 | 2,2,2-trifluoroacetamide |
| BAY-1251152-007 | 1610359-06-2 | (E)-2,2,2-trifluoro-N-(((2-((5-fluoro-4-(4-fluoro-2-methoxyphenyl)pyridin-2-yl)amino)pyridin-4-yl)methyl)(methyl)-l4-sulfaneylidene)acetamide |
Frequently asked questions
What are the approved indications of Enitociclib?
Approved indications include: Non-Hodgkin lymphoma, Lymphoma, Haematological malignancy, Neoplasm, 里氏综合征, Chronic lymphocytic leukaemia.
When does the Enitociclib patent expire?
No public expiry year is available for Enitociclib yet; this page updates once verified.
How many synthesis routes are recorded for Enitociclib?
1 synthesis routes are recorded; the shortest is 4 steps with 50 mg (BAY-1251152) total yield. Intermediates in each route carry codes and CAS numbers.
Where can I buy Enitociclib intermediates?
All intermediates in Enitociclib routes have CAS profiles — you can submit an RFQ per CAS and it enters the Unibest matching pool.
How do I get a quote for Enitociclib intermediates?
Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.
Source: cross-verified data (structured fields only) · 2026-10-22